WLB-89462

WLB-89462 : Modulator of TMEM97

Structure

Information

  • TMEM97
  • Modulator
  • up to 1 uM

In Vitro Validations

No in Vitro Validations

In Cell Validations

In Vivo Data

Off-Target Selectivity Assesments

Potency assay (off target): Highly selective vs both the σ1R (IC50 1777 nM) and a general panel of 180 different targets, composed different receptors, ion channels and transporters (Eurofins), showing no no target inhibition above 50% with screening at 10 μM
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SERP ratings and comments


No SERP comments found for WLB-89462